()-N6-(2-Phenylisopropyl)adenosine

About ()-N6-(2-Phenylisopropyl)adenosine

()-N6-(2-Phenylisopropyl)adenosine Synonym: (R)-N6-(1-Methyl-2-phenylethyl)adenosine, N6-(L-2-Phenylisopropyl)adenosine, R-()-PIA Empirical Formula (Hill Notation): C19H23N5O4Molecular Weight: 385.42CAS Number: 38594-96-6 form solid potency 1.17nM Ki for A1 receptors (using [3H]CHA in rat forebrain preparations) color white solubility H2O: slightly soluble0.3mg/mL (Solutions may be stored for several days at 4C.) 45% (w/v) aq 2-hydroxypropyl--cyclodextrin: soluble1.6mg/mL (Solutions may be stored for several days at 4C.) storage temp. 2-8C Gene Information human ... ADORA1(134) Description Packaging 25 mg in poly bottle 50, 100 mg in glass bottle Biochem/physiol Actions A1 adenosine receptor agonist. Affinity for adenosine receptor is approx. 100 that of the (+)-isomer. Features and Benefits This compound is also offered as part of Sigmas Library of Pharmacologically Active Compounds (LOPAC1280), a biologically annotated collection of high-quality, ready-to-screen compounds. This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction.